Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Casein kinase I isoform alpha (Homo sapiens (Human)) | BDBM50260229 (4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-im...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto di Ricerche di Biologia Molecolare "P. Angeletti Curated by ChEMBL | Assay Description Inhibition of human CKIalpha | J Biol Chem 282: 5536-44 (2007) Article DOI: 10.1074/jbc.M610486200 BindingDB Entry DOI: 10.7270/Q2M32VJH | |||||||||||
More data for this Ligand-Target Pair |