Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Chloroquine resistance transporter (Plasmodium falciparum) | BDBM50017696 ((2-dimethylamino-2-methyl)ethyl-N-dibenzoparathiaz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 8.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Australian National University Curated by ChEMBL | Assay Description Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c... | ACS Med Chem Lett 5: 576-81 (2014) Article DOI: 10.1021/ml5000228 BindingDB Entry DOI: 10.7270/Q22V2HPS | |||||||||||
More data for this Ligand-Target Pair |