Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholesteryl ester transfer protein (Homo sapiens (Human)) | BDBM50070315 ((3S,9S)-9-Benzyl-3-isobutyl-6-methyl-13-(1-methyl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering Plough Research Institute Curated by ChEMBL | Assay Description Compound was evaluated for inhibitory activity against cholesteryl ester transfer protein | Bioorg Med Chem Lett 8: 1277-80 (1999) BindingDB Entry DOI: 10.7270/Q25X282F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholesteryl ester transfer protein (Homo sapiens (Human)) | BDBM50070315 ((3S,9S)-9-Benzyl-3-isobutyl-6-methyl-13-(1-methyl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering Plough Research Institute Curated by ChEMBL | Assay Description Tested for inhibition of substrate hydrolysis in the presence of porcine kidney esterase at a concentration of 45 nM | Bioorg Med Chem Lett 8: 1277-80 (1999) BindingDB Entry DOI: 10.7270/Q25X282F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholesteryl ester transfer protein (Homo sapiens (Human)) | BDBM50070315 ((3S,9S)-9-Benzyl-3-isobutyl-6-methyl-13-(1-methyl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering Plough Research Institute Curated by ChEMBL | Assay Description pA2 value towards endothelin receptor A was determined as functional ETA antagonism | Bioorg Med Chem Lett 8: 1277-80 (1999) BindingDB Entry DOI: 10.7270/Q25X282F | |||||||||||
More data for this Ligand-Target Pair |