Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50009070 ((2S,3R)-3-(2-Carboxy-ethylsulfanyl)-2-hydroxy-3-[2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displasement of [3H]-LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50009070 ((2S,3R)-3-(2-Carboxy-ethylsulfanyl)-2-hydroxy-3-[2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-LTD4 from LTD4 receptor in guinea pig lung membranes | J Med Chem 34: 1235-42 (1991) BindingDB Entry DOI: 10.7270/Q2K936HB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50009070 ((2S,3R)-3-(2-Carboxy-ethylsulfanyl)-2-hydroxy-3-[2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity against Cysteinyl leukotriene D4 receptor in guinea pig lung membranes using [3H]-LTD4 as the radioligand. | J Med Chem 30: 959-61 (1987) BindingDB Entry DOI: 10.7270/Q2D50KZN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (Homo sapiens (Human)) | BDBM50009070 ((2S,3R)-3-(2-Carboxy-ethylsulfanyl)-2-hydroxy-3-[2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity against Cysteinyl leukotriene D4 receptor in guinea pig lung membranes using [3H]-LTD4 as the radioligand. | J Med Chem 30: 959-61 (1987) BindingDB Entry DOI: 10.7270/Q2D50KZN | |||||||||||
More data for this Ligand-Target Pair |