Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50313915 (2,8,9,13b-Tetrahydro-6H-isoquino[2,1-b]pyrrolo[4,3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Schiller-Universit£t Jena Curated by ChEMBL | Assay Description Displacement of [3H]radioligand from human recombinant dopamine D3 receptor expressed in HEK293 cells by microplate scintillation counting | J Med Chem 53: 2646-50 (2010) Article DOI: 10.1021/jm901291r BindingDB Entry DOI: 10.7270/Q2SJ1KRJ | |||||||||||
More data for this Ligand-Target Pair |