BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM50306287'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50306287 (3-(4-(4-(3-hydroxypentan-3-yl)phenyl)-1-(2-methylp...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Pfizer Global Research and Development Curated by ChEMBL					Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting				Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1
Pfizer Global Research and Development Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50306287 (3-(4-(4-(3-hydroxypentan-3-yl)phenyl)-1-(2-methylp...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.70	n/a	n/a	n/a	n/a	n/a	n/a
Pfizer Global Research and Development Curated by ChEMBL					Assay Description Antagonist activity at delta opioid receptor by GTPgammaS bunding assay				Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1
Pfizer Global Research and Development Curated by ChEMBL					More data for this Ligand-Target Pair