Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dopamine receptors; D2 & D4 (Homo sapiens (Human)) | BDBM50027079![]() (CHEMBL3335539) | Reactome pathway KEGG DrugBank GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Inhibition of human dopamine D4 receptor | ACS Med Chem Lett 5: 1060-4 (2014) Article DOI: 10.1021/ml500267c BindingDB Entry DOI: 10.7270/Q2G44RWM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dopamine receptors; D2 & D4 (Homo sapiens (Human)) | BDBM50027079![]() (CHEMBL3335539) | Reactome pathway KEGG DrugBank GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Inhibition of human dopamine D4 receptor | ACS Med Chem Lett 5: 1060-4 (2014) Article DOI: 10.1021/ml500267c BindingDB Entry DOI: 10.7270/Q2G44RWM | |||||||||||
More data for this Ligand-Target Pair |