Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ELAV-like protein 1 (Homo sapiens (Human)) | BDBM50326009 (5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein interaction with TMR-labeled A/U-rich element of TNFalpha by confocal fluctuation ... | Nat Chem Biol 3: 508-15 (2007) Article DOI: 10.1038/nchembio.2007.14 BindingDB Entry DOI: 10.7270/Q2QN670V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ELAV-like protein 1 (Homo sapiens (Human)) | BDBM50326009 (5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein dimerization with TMR-labeled A/U-rich element of IL-2 by confocal fluctuation spe... | Nat Chem Biol 3: 508-15 (2007) Article DOI: 10.1038/nchembio.2007.14 BindingDB Entry DOI: 10.7270/Q2QN670V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ELAV-like protein 1 (Homo sapiens (Human)) | BDBM50326009 (5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein dimerization with TMR-labeled A/U-rich element of TNFalpha by confocal fluctuation... | Nat Chem Biol 3: 508-15 (2007) Article DOI: 10.1038/nchembio.2007.14 BindingDB Entry DOI: 10.7270/Q2QN670V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ELAV-like protein 1 (Homo sapiens (Human)) | BDBM50326009 (5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Binding affinity recombinant HuR RRM1/RRM2 domain by confocal fluctuation spectroscopy | Nat Chem Biol 3: 508-15 (2007) Article DOI: 10.1038/nchembio.2007.14 BindingDB Entry DOI: 10.7270/Q2QN670V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ELAV-like protein 1 (Homo sapiens (Human)) | BDBM50326009 (5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein interaction with TMR-labeled A/U-rich element of IL-2 by confocal fluctuation spec... | Nat Chem Biol 3: 508-15 (2007) Article DOI: 10.1038/nchembio.2007.14 BindingDB Entry DOI: 10.7270/Q2QN670V | |||||||||||
More data for this Ligand-Target Pair |