Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2 (Homo sapiens (Human)) | BDBM50110402 (CHEMBL3605581) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.79E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Georgia Curated by ChEMBL | Assay Description Inhibition of human ATX phosphodiesterase expressed in Sf9 cells assessed as hydrolysis of FS-3 measured after 5 to 25 mins by fluorescence assay | Bioorg Med Chem 23: 5999-6013 (2015) Article DOI: 10.1016/j.bmc.2015.06.054 BindingDB Entry DOI: 10.7270/Q2K9399W | |||||||||||
More data for this Ligand-Target Pair |