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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Ephrin type-B receptor 3 (EPHB3)' and Ligand = 'BDBM50311304'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Ephrin type-B receptor 3 (EPHB3)


(Homo sapiens (Human))
BDBM50311304
PNG
(CHEMBL1078108 | N-(2-chlorophenyl)-5-(1H-pyrrol-1-...)
Show SMILES Clc1ccccc1NC(=O)c1cnn2ccc(cc12)-n1cccc1
Show InChI InChI=1S/C18H13ClN4O/c19-15-5-1-2-6-16(15)21-18(24)14-12-20-23-10-7-13(11-17(14)23)22-8-3-4-9-22/h1-12H,(H,21,24)
PDB
MMDB

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PC cid
PC sid
UniChem
Article
PubMed
n/an/a 200n/an/an/an/an/an/a



Harvard Medical School

Curated by ChEMBL


Assay Description
Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...


Bioorg Med Chem Lett 19: 6122-6 (2009)


Article DOI: 10.1016/j.bmcl.2009.09.010
BindingDB Entry DOI: 10.7270/Q2T43T66
More data for this
Ligand-Target Pair