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Found 1 hit Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM19453'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Estrogen receptor


(Homo sapiens (Human))		BDBM19453
PNG
(4-[3-phenyl-5,7-bis(trifluoromethyl)pyrazolo[1,5-a...)
Show SMILES Oc1ccc(cc1)-c1nn2c(cc(nc2c1-c1ccccc1)C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C20H11F6N3O/c21-19(22,23)14-10-15(20(24,25)26)29-18(27-14)16(11-4-2-1-3-5-11)17(28-29)12-6-8-13(30)9-7-12/h1-10,30H
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars
Article
PubMed
 51 -38.1n/an/an/an/an/a7.50



University of Illinois at Urbana



Assay Description
Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...

J Med Chem 50: 399-403 (2007)


Article DOI: 10.1021/jm061035y
BindingDB Entry DOI: 10.7270/Q2QZ288F
More data for this
Ligand-Target Pair