Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Eukaryotic translation initiation factor 2-alpha kinase 1 (Homo sapiens (Human)) | BDBM50072073 (CHEMBL3407848) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of HRI (unknown origin) | J Med Chem 58: 1426-41 (2015) Article DOI: 10.1021/jm5017494 BindingDB Entry DOI: 10.7270/Q27W6DWN | |||||||||||
More data for this Ligand-Target Pair |