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Found 1 hit Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 4' and Ligand = 'BDBM50437959'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
G protein-activated inward rectifier potassium channel 4


(Homo sapiens (Human))
BDBM50437959
PNG
(CHEMBL2409123)
Show SMILES CC(C)c1cc(NC(=O)Nc2cccc(c2)C(F)(F)F)n(n1)-c1ccccc1
Show InChI InChI=1S/C20H19F3N4O/c1-13(2)17-12-18(27(26-17)16-9-4-3-5-10-16)25-19(28)24-15-8-6-7-14(11-15)20(21,22)23/h3-13H,1-2H3,(H2,24,25,28)
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PC cid
PC sid
UniChem
Article
PubMed
n/an/a 1.30E+3n/an/an/an/an/an/a



Northwest Agriculture& Forestry University

Curated by ChEMBL


Assay Description
Inhibition of GIRK1/4 (unknown origin)


Bioorg Med Chem Lett 23: 4562-6 (2013)


Article DOI: 10.1016/j.bmcl.2013.06.023
More data for this
Ligand-Target Pair