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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50433580'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucagon receptor


(Homo sapiens (Human))		BDBM50433580
PNG
(CHEMBL2381844)
Show SMILES CCCC(Oc1ccc(cc1)-n1cc(cn1)C(=O)N(C)C)c1ccc(cc1)C(=O)NCCC(O)=O
Show InChI InChI=1S/C26H30N4O5/c1-4-5-23(18-6-8-19(9-7-18)25(33)27-15-14-24(31)32)35-22-12-10-21(11-13-22)30-17-20(16-28-30)26(34)29(2)3/h6-13,16-17,23H,4-5,14-15H2,1-3H3,(H,27,33)(H,31,32)
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PC cid
PC sid
UniChem

Similars
Article
PubMed
 6.50E+3n/an/an/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Displacement of [125I]-glucagon-cex from human glucagon receptor by cell based assay in presence of 0.2% bovine serum albumin

Bioorg Med Chem Lett 23: 3051-8 (2013)


Article DOI: 10.1016/j.bmcl.2013.03.014
BindingDB Entry DOI: 10.7270/Q27M099R
More data for this
Ligand-Target Pair