Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50412519 (CHEMBL455662) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.16 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Binding affinity to glucocorticoid receptor | Bioorg Med Chem Lett 18: 6097-9 (2008) Article DOI: 10.1016/j.bmcl.2008.10.021 BindingDB Entry DOI: 10.7270/Q2668FDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50412519 (CHEMBL455662) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Agonist activity at glucocorticoid receptor by MMTV transactivation assay | Bioorg Med Chem Lett 18: 6097-9 (2008) Article DOI: 10.1016/j.bmcl.2008.10.021 BindingDB Entry DOI: 10.7270/Q2668FDB | |||||||||||
More data for this Ligand-Target Pair |