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Found 1 hit Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 2' and Ligand = 'BDBM50088227'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glutamate receptor ionotropic, kainate 2


(Homo sapiens (Human))		BDBM50088227
PNG
(CHEMBL58054 | E-2-Amino-4-[3-(3-chloro-phenyl)-all...)
Show SMILES N[C@@H](C[C@@H](C\C=C\c1cccc(Cl)c1)C(O)=O)C(O)=O
Show InChI InChI=1S/C14H16ClNO4/c15-11-6-2-4-9(7-11)3-1-5-10(13(17)18)8-12(16)14(19)20/h1-4,6-7,10,12H,5,8,16H2,(H,17,18)(H,19,20)/b3-1+/t10-,12+/m1/s1
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PubMed
 1.13E+3n/an/an/an/an/an/an/an/a



Lilly, S.A.

Curated by ChEMBL


Assay Description
Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]-kainate as radioligand

J Med Chem 43: 1958-68 (2000)


BindingDB Entry DOI: 10.7270/Q2FX78QB
More data for this
Ligand-Target Pair