Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Heparanase (Homo sapiens (Human)) | BDBM50307388 (8-(4-Phenyl[1,2,3]triazol-1-yl)octyl 2,3,4,6-Tetra...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a |
Progen Pharmaceuticals Limited Curated by ChEMBL | Assay Description Inhibition of human recombinant heparanase | J Med Chem 53: 1686-99 (2010) Article DOI: 10.1021/jm901449m BindingDB Entry DOI: 10.7270/Q2PG1SPH | |||||||||||
More data for this Ligand-Target Pair |