Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM50131679 (CHEMBL3628211 | p-Hydroxyphenylethyl p-coumarate (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.02E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His-tagged cytoplasmic c-MET kinase domain (956 to 1390 residues) phosphorylation expressed in baculovirus... | Eur J Med Chem 118: 299-315 (2016) Article DOI: 10.1016/j.ejmech.2016.04.043 BindingDB Entry DOI: 10.7270/Q2GT5Q35 | |||||||||||
More data for this Ligand-Target Pair |