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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histamine H1 receptor' and Ligand = 'BDBM50002101'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H1 receptor


(Cavia porcellus (domestic guinea pig))		BDBM50002101
PNG
(11-(2-Dimethylamino-ethylidene)-6,11-dihydro-diben...)
Show SMILES CN(C)C\C=C1/c2ccccc2COc2ccc(cc12)C(O)=O
Show InChI InChI=1S/C19H19NO3/c1-20(2)10-9-16-15-6-4-3-5-14(15)12-23-18-8-7-13(19(21)22)11-17(16)18/h3-9,11H,10,12H2,1-2H3,(H,21,22)/b16-9+
UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
 12n/an/an/an/an/an/an/an/a



Kyowa Hakko Kogyo Co., Ltd.

Curated by ChEMBL


Assay Description
Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uM

J Med Chem 35: 2074-84 (1992)


BindingDB Entry DOI: 10.7270/Q2N87BC0
More data for this
Ligand-Target Pair