Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50070217 (3-(3-Bromo-4-methoxy-phenyl)-2-[(E)-hydroxyimino]-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Gliatech Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptor | Bioorg Med Chem Lett 8: 1133-8 (1999) BindingDB Entry DOI: 10.7270/Q2GF0SPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (GUINEA PIG) | BDBM50070217 (3-(3-Bromo-4-methoxy-phenyl)-2-[(E)-hydroxyimino]-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to histamine H3 receptor in guinea pig brain membrane | J Nat Prod 57: 175-177 (1994) Article DOI: 10.1021/np50103a029 BindingDB Entry DOI: 10.7270/Q2ZK5GPT | |||||||||||
More data for this Ligand-Target Pair |