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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50092855'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Rattus norvegicus (rat))		BDBM50092855
PNG
(CHEMBL129146 | Cyclopentyl-{4-[3-(1H-imidazol-4-yl...)
Show SMILES O=C(C1CCCC1)c1ccc(OCCCc2cnc[nH]2)cc1
Show InChI InChI=1S/C18H22N2O2/c21-18(14-4-1-2-5-14)15-7-9-17(10-8-15)22-11-3-6-16-12-19-13-20-16/h7-10,12-14H,1-6,11H2,(H,19,20)
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Similars
PubMed
 7.20n/an/an/an/an/an/an/an/a



Freie Universit£t Berlin

Curated by ChEMBL


Assay Description
Effect on histamine H3 receptors in vitro, on synaptosomes of rat cerebral cortex for the release of [3H]histamine

J Med Chem 43: 3987-94 (2000)


BindingDB Entry DOI: 10.7270/Q2833SRN
More data for this
Ligand-Target Pair