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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50092862'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Rattus norvegicus (rat))		BDBM50092862
PNG
(5-[3-(1H-Imidazol-4-yl)-propoxy]-indan-1-one; comp...)
Show SMILES O=C1CCc2cc(OCCCc3cnc[nH]3)ccc12
Show InChI InChI=1S/C15H16N2O2/c18-15-6-3-11-8-13(4-5-14(11)15)19-7-1-2-12-9-16-10-17-12/h4-5,8-10H,1-3,6-7H2,(H,16,17)
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PubMed
 17n/an/an/an/an/an/an/an/a



Freie Universit£t Berlin

Curated by ChEMBL


Assay Description
Compounds were tested for their effect at histamine H3 receptors in vitro on synaptosomes of rat cerebral cortex for the release of [3H]histamine

J Med Chem 43: 3987-94 (2000)


BindingDB Entry DOI: 10.7270/Q2833SRN
More data for this
Ligand-Target Pair