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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50093225'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Rattus norvegicus (rat))		BDBM50093225
PNG
(CHEMBL76440 | Cyclopropyl-{4-[2-(1H-imidazol-4-yl)...)
Show SMILES O=C(C1CC1)c1ccc(OCCc2cnc[nH]2)cc1
Show InChI InChI=1S/C15H16N2O2/c18-15(11-1-2-11)12-3-5-14(6-4-12)19-8-7-13-9-16-10-17-13/h3-6,9-11H,1-2,7-8H2,(H,16,17)
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Similars
PubMed
 2.10n/an/an/an/an/an/an/an/a



Freie Universität Berlin

Curated by ChEMBL


Assay Description
In vitro inhibitory activity against Histamine H3 receptor for K+ evoked depolarization-induced release of [3H]-histamine from synaptosomes of rat ce...

Bioorg Med Chem Lett 10: 2379-82 (2001)


BindingDB Entry DOI: 10.7270/Q28G8JZ4
More data for this
Ligand-Target Pair