BindingDB PrimarySearch

Found 1 hit Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT5' and Ligand = 'BDBM50255522'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Histone acetyltransferase KAT5 (Homo sapiens (Human))	BDBM50255522 (Ac-ARTKQTARKSTGGK(CoA)APRKQL \| CHEMBL526343) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.96E+4	n/a	n/a	n/a	n/a	n/a	n/a
Georgia State University Curated by ChEMBL					Assay Description Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillation				Bioorg Med Chem 17: 1381-6 (2009) Article DOI: 10.1016/j.bmc.2008.12.014 BindingDB Entry DOI: 10.7270/Q2K35VKS
Georgia State University Curated by ChEMBL					More data for this Ligand-Target Pair