Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig)) | BDBM50033143 (CHEMBL216640 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.580 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593 | J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q | |||||||||||
More data for this Ligand-Target Pair |