Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Kappa-type opioid receptor (Mus musculus (Mouse)) | BDBM50120877 (2-[(2-{5-Guanidino-2-[3-(3-hydroxy-phenyl)-2-methy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Daiichi Fine Chemical Co. Ltd. Curated by ChEMBL | Assay Description Binding affinity of the compound towards Opioid receptor kappa 1 by the displacement of [3H]-U-69,593 in mouse spinal cord | J Med Chem 45: 5081-9 (2002) BindingDB Entry DOI: 10.7270/Q290233R | |||||||||||
More data for this Ligand-Target Pair |