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Found 1 hit Enz. Inhib. hit(s) with Target = 'Leucine aminopeptidase (LAP)' and Ligand = 'BDBM234298'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Leucine aminopeptidase (LAP)


(Sus scrofa (Pig))
BDBM234298
PNG
(Nle-ψ[P(O)(OH)O]-L-Ala (6))
Show SMILES CCCCC(N)P(O)(=O)O[C@@H](C)C(O)=O |r|
Show InChI InChI=1/C8H18NO5P/c1-3-4-5-7(9)15(12,13)14-6(2)8(10)11/h6-7H,3-5,9H2,1-2H3,(H,10,11)(H,12,13)/t6-,7?/s2
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
2.69E+5 -20.4n/an/an/an/an/a8.425



Academy of Sciences of the Czech Republic



Assay Description
LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25C. The substrate (L-leucine-p-nitroanilide) was...


J Enzyme Inhib Med Chem 26: 155-61 (2011)


Article DOI: 10.3109/14756366.2010.482047
More data for this
Ligand-Target Pair