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Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 2B' and Ligand = 'BDBM319653'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Lysine-specific demethylase 2B


(Homo sapiens (Human))		BDBM319653
PNG
(2-(1-benzyl-1H-imidazol-4-yl)-4-[5- (trifluorometh...)
Show SMILES FC(F)(F)c1[nH]nnc1-c1ccnc(c1)-c1cn(Cc2ccccc2)cn1
Show InChI InChI=1S/C18H13F3N6/c19-18(20,21)17-16(24-26-25-17)13-6-7-22-14(8-13)15-10-27(11-23-15)9-12-4-2-1-3-5-12/h1-8,10-11H,9H2,(H,24,25,26)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



GSK



Assay Description
The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...

Bioorg Med Chem Lett 17: 1584-9 (2007)


BindingDB Entry DOI: 10.7270/Q2FT8PBQ
More data for this
Ligand-Target Pair