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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4C' and Ligand = 'BDBM277750'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Lysine-specific demethylase 4C


(Homo sapiens (Human))		BDBM277750
PNG
(3-({5-fluoro-1-[2-(piperidin-3-yl)ethyl]-1H-indazo...)
Show SMILES OC(=O)c1ccncc1Nc1nn(CCC2CCCNC2)c2ccc(F)cc12
Show InChI InChI=1S/C20H22FN5O2/c21-14-3-4-18-16(10-14)19(24-17-12-23-8-5-15(17)20(27)28)25-26(18)9-6-13-2-1-7-22-11-13/h3-5,8,10,12-13,22H,1-2,6-7,9,11H2,(H,24,25)(H,27,28)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Celgene Quanticel Research Inc

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...

US Patent US10336727 (2019)


BindingDB Entry DOI: 10.7270/Q2571FBT
More data for this
Ligand-Target Pair