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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4C' and Ligand = 'BDBM347129'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Lysine-specific demethylase 4C


(Homo sapiens (Human))		BDBM347129
PNG
(-(4-(methyl(3-(4-methylpiperazin-1-yl)-4- (2,2,2-t...)
Show SMILES CN(c1ccc(Oc2nc(O)c3ccncc3n2)cc1)c1ccc(OCC(F)(F)F)c(c1)N1CCN(C)CC1
Show InChI InChI=1S/C27H27F3N6O3/c1-34-11-13-36(14-12-34)23-15-19(5-8-24(23)38-17-27(28,29)30)35(2)18-3-6-20(7-4-18)39-26-32-22-16-31-10-9-21(22)25(37)33-26/h3-10,15-16H,11-14,17H2,1-2H3,(H,32,33,37)
PDB

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US Patent
n/an/a<100n/an/an/an/an/an/a



CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...

US Patent US10202381 (2019)


BindingDB Entry DOI: 10.7270/Q2SX6GBM
More data for this
Ligand-Target Pair