Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lysine-specific demethylase 5A (Homo sapiens (Human)) | BDBM154552 (N1-(3-Bromobenzyl)-N3-(tert-butyl)propane-1,3-diam...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | 8.0 | 1,390.75 |
University of North Carolina at Chapel Hill | Assay Description In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ... | ACS Chem Biol 10: 1072-81 (2015) Article DOI: 10.1021/cb500956g BindingDB Entry DOI: 10.7270/Q27S7MHJ | |||||||||||
More data for this Ligand-Target Pair |