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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific histone demethylase 1A' and Ligand = 'BDBM179724'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Lysine-specific histone demethylase 1A


(Homo sapiens (Human))
BDBM179724
PNG
(US9676701, 46 5-(5-((trans)-2-aminocyclopropyl)pyr...)
Show SMILES Cc1ccc(cc1O)-c1ccc(cn1)[C@H]1C[C@@H]1N |r|
Show InChI InChI=1/C15H16N2O/c1-9-2-3-10(6-15(9)18)14-5-4-11(8-17-14)12-7-13(12)16/h2-6,8,12-13,18H,7,16H2,1H3/t12-,13+/s2
PDB
MMDB

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KEGG

UniProtKB/SwissProt

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antibodypedia
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PC cid
PC sid
UniChem
US Patent
50 -41.7n/an/an/an/an/a7.425



ORYZON GENOMICS, S.A.

US Patent


Assay Description
Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of various concentrations of inhibitor (e....


US Patent US9676701 (2017)


BindingDB Entry DOI: 10.7270/Q27P8WJN
More data for this
Ligand-Target Pair