Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Macrophage-stimulating protein receptor (Homo sapiens (Human)) | BDBM50317324 (CHEMBL1087984 | N-(4-(6,7-dimethoxyquinolin-4-ylox...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
ChemRF Laboratories Curated by ChEMBL | Assay Description Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISA | Bioorg Med Chem Lett 25: 2527-31 (2015) Article DOI: 10.1016/j.bmcl.2015.04.056 BindingDB Entry DOI: 10.7270/Q21C1ZMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Macrophage-stimulating protein receptor (Homo sapiens (Human)) | BDBM50317324 (CHEMBL1087984 | N-(4-(6,7-dimethoxyquinolin-4-ylox...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
MethylGene Inc. Curated by ChEMBL | Assay Description Inhibition of TPR-tagged RON catalytic domain expressed in HEK293 cells | Bioorg Med Chem Lett 20: 2745-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.073 BindingDB Entry DOI: 10.7270/Q24T6JJ6 | |||||||||||
More data for this Ligand-Target Pair |