BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50168509'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Melanin-concentrating hormone receptor 1 (Mus musculus)	BDBM50168509 (CHEMBL188937 \| N-(1-Benzo[1,3]dioxol-5-ylmethyl-pi...) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Abbott Laboratories Curated by ChEMBL					Assay Description Inhibitory concentration required for binding affinity against mouse MCHr1 competing human neuronal IMR32 cells receptor in a radiometric binding ass...				Bioorg Med Chem Lett 15: 3412-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.023 BindingDB Entry DOI: 10.7270/Q26D5SHR
Abbott Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Melanin-concentrating hormone receptor 1 (Mus musculus)	BDBM50168509 (CHEMBL188937 \| N-(1-Benzo[1,3]dioxol-5-ylmethyl-pi...) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	90	n/a	n/a	n/a	n/a	n/a	n/a
Abbott Laboratories Curated by ChEMBL					Assay Description Inhibitory concentration required for functional antagonism of MCH mediated Ca+2 release competing human IMR32 cells receptor in a FLIPRTM based assa...				Bioorg Med Chem Lett 15: 3412-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.023 BindingDB Entry DOI: 10.7270/Q26D5SHR
Abbott Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair