Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 4 (Mus musculus) | BDBM50166123 (CHEMBL408600 | [(2S,5R,8R,11R,14S,17R)-1-(2-Acetyl...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0600 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description In vitro agonist potency for Mouse Melanocortin 4 receptor | J Med Chem 48: 3328-36 (2005) Article DOI: 10.1021/jm0490843 BindingDB Entry DOI: 10.7270/Q29K4C0B | |||||||||||
More data for this Ligand-Target Pair |