BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50189010'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Melanocortin receptor 4 (Homo sapiens (Human))	BDBM50189010 ((S)-2-[(S)-4-{(R)-2-[(S)-2-acetylamino-3-(4-hydrox...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	0.600	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Procter & Gamble Pharmaceuticals Curated by ChEMBL					Assay Description Binding affinity to human MC4R				Bioorg Med Chem Lett 16: 4668-73 (2006) Article DOI: 10.1016/j.bmcl.2006.05.087 BindingDB Entry DOI: 10.7270/Q2W66KDF
Procter & Gamble Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Melanocortin receptor 4 (Homo sapiens (Human))	BDBM50189010 ((S)-2-[(S)-4-{(R)-2-[(S)-2-acetylamino-3-(4-hydrox...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	0.200	n/a	n/a	n/a	n/a
Procter & Gamble Pharmaceuticals Curated by ChEMBL					Assay Description Agonist activity at human MC4R				Bioorg Med Chem Lett 16: 4668-73 (2006) Article DOI: 10.1016/j.bmcl.2006.05.087 BindingDB Entry DOI: 10.7270/Q2W66KDF
Procter & Gamble Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair