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Found 1 hit Enz. Inhib. hit(s) with Target = 'Microtubule-associated protein 2' and Ligand = 'BDBM50234021'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Microtubule-associated protein 2


(Homo sapiens (Human))
BDBM50234021
PNG
(CHEMBL4074903)
Show SMILES Fc1cccc(OC[C@H]2CCCN2c2ncnc3[nH]cnc23)c1 |r|
Show InChI InChI=1S/C16H16FN5O/c17-11-3-1-5-13(7-11)23-8-12-4-2-6-22(12)16-14-15(19-9-18-14)20-10-21-16/h1,3,5,7,9-10,12H,2,4,6,8H2,(H,18,19,20,21)/t12-/m1/s1
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 2.00E+3n/an/an/an/an/an/a



Merck KGaA

Curated by ChEMBL


Assay Description
Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...


Bioorg Med Chem Lett 27: 551-556 (2017)


Article DOI: 10.1016/j.bmcl.2016.12.019
BindingDB Entry DOI: 10.7270/Q2V98BB4
More data for this
Ligand-Target Pair