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Found 1 hit Enz. Inhib. hit(s) with Target = 'Microtubule-associated protein 2' and Ligand = 'BDBM50435183'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Microtubule-associated protein 2


(Homo sapiens (Human))		BDBM50435183
PNG
(CHEMBL2392933)
Show SMILES Cc1nc(nc(NCC(CCCc2ccccc2)c2ccccc2)c1Cl)-c1ccc(Cl)cn1
Show InChI InChI=1S/C27H26Cl2N4/c1-19-25(29)27(33-26(32-19)24-16-15-23(28)18-30-24)31-17-22(21-12-6-3-7-13-21)14-8-11-20-9-4-2-5-10-20/h2-7,9-10,12-13,15-16,18,22H,8,11,14,17H2,1H3,(H,31,32,33)
KEGG

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PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a>2.00E+5n/an/an/an/a



Chinese Academy of Sciences

Curated by ChEMBL


Assay Description
Inhibition of human recombinant GST-6XHis-tagged full-length cytosolic METAP2 expressed in cabbage looper BTI-TN-5B1-4 cells using Met-Pro-p-nitroani...

Bioorg Med Chem 21: 2600-17 (2013)


Article DOI: 10.1016/j.bmc.2013.02.023
BindingDB Entry DOI: 10.7270/Q290256X
More data for this
Ligand-Target Pair