Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mitogen-activated protein kinase kinase kinase 11 (Homo sapiens (Human)) | BDBM50108291 (CHEMBL36891 | Indolocarbazole analogue) | PDB NCI pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyowa-Hakko Kogyo Co., Ltd. Curated by ChEMBL | Assay Description Inhibition of Mixed lineage kinase 3 (MLK3) | Bioorg Med Chem Lett 12: 147-50 (2001) BindingDB Entry DOI: 10.7270/Q2571B94 | |||||||||||
More data for this Ligand-Target Pair |