Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50127701 (CHEMBL3627737) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.515 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lanzhou University Curated by ChEMBL | Assay Description Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) transfected in HEK293 cells | Bioorg Med Chem Lett 25: 5393-7 (2015) Article DOI: 10.1016/j.bmcl.2015.09.025 BindingDB Entry DOI: 10.7270/Q24M96CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50127701 (CHEMBL3627737) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0643 | n/a | n/a | n/a | n/a |
Lanzhou University Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor (unknown origin) transfected in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP production | Bioorg Med Chem Lett 25: 5393-7 (2015) Article DOI: 10.1016/j.bmcl.2015.09.025 BindingDB Entry DOI: 10.7270/Q24M96CW | |||||||||||
More data for this Ligand-Target Pair |