BindingDB PrimarySearch

Found 3 hits Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50240679'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mu-type opioid receptor (Rattus norvegicus (rat))	BDBM50240679 (2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-(3-hyd...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	151	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Cagliary Curated by ChEMBL					Assay Description Binding affinity for rat brain P2 synaptosome Opioid receptor mu 1				J Med Chem 45: 713-20 (2002) BindingDB Entry DOI: 10.7270/Q2639QFF
University of Cagliary Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50240679 (2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-(3-hyd...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	151	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Naples Curated by ChEMBL					Assay Description Inhibition of guinea pig ileum Opioid receptor mu 1				Bioorg Med Chem Lett 10: 2745-8 (2000) BindingDB Entry DOI: 10.7270/Q25H7HF1
University of Naples Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50240679 (2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-(3-hyd...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	n/a	n/a	<1.00E+4	n/a	n/a	n/a	n/a
University of Naples Curated by ChEMBL					Assay Description Negative logarithm of the molar concentration for agonist activity at Opioid receptor mu 1 was determined in guinea pig ileum				Bioorg Med Chem Lett 10: 2745-8 (2000) BindingDB Entry DOI: 10.7270/Q25H7HF1
University of Naples Curated by ChEMBL					More data for this Ligand-Target Pair