Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50092313 (1-Cyclohexyl-4-{1-[4-(4-methoxy-benzenesulfinyl)-p...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.530 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Binding affinity against Muscarinic acetylcholine receptor M1 | Bioorg Med Chem Lett 10: 2209-12 (2001) BindingDB Entry DOI: 10.7270/Q24T6HMP | |||||||||||
More data for this Ligand-Target Pair |