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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50326238'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Muscarinic acetylcholine receptor M1


(Homo sapiens (Human))		BDBM50326238
PNG
(CHEMBL1243109 | N-{1-[3-(7-Methoxy-2-oxo-3,4-dihyd...)
Show SMILES COc1ccc2CCC(=O)N(CCCN3CCC(CC3)NC(=O)Cc3ccccc3)c2c1
Show InChI InChI=1S/C26H33N3O3/c1-32-23-10-8-21-9-11-26(31)29(24(21)19-23)15-5-14-28-16-12-22(13-17-28)27-25(30)18-20-6-3-2-4-7-20/h2-4,6-8,10,19,22H,5,9,11-18H2,1H3,(H,27,30)
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Similars
Article
PubMed
n/an/an/an/a 120n/an/an/an/a



H. Lundbeck A/S

Curated by ChEMBL


Assay Description
Agonist activity at human muscarinic M1 receptor expressed in CHO-K1 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assay

J Med Chem 53: 6386-97 (2010)


Article DOI: 10.1021/jm100697g
BindingDB Entry DOI: 10.7270/Q2765G9K
More data for this
Ligand-Target Pair