Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M1 (RAT) | BDBM50356966 (CHEMBL1916224) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 110 | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Agonist activity at rat muscarinic M1 receptor expressed in CHO cells | Bioorg Med Chem Lett 21: 6451-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.084 BindingDB Entry DOI: 10.7270/Q26W9BG8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50356966 (CHEMBL1916224) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 890 | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Agonist activity at human muscarinic M1 receptor | Bioorg Med Chem Lett 22: 3467-72 (2012) Article DOI: 10.1016/j.bmcl.2012.03.088 BindingDB Entry DOI: 10.7270/Q28916WQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (RAT) | BDBM50356966 (CHEMBL1916224) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Agonist activity at rat recombinant muscarinic M1 receptor by HTS cell based assay | Bioorg Med Chem Lett 21: 6451-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.084 BindingDB Entry DOI: 10.7270/Q26W9BG8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50356966 (CHEMBL1916224) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Agonist activity at human recombinant muscarinic M1 receptor by HTS cell based assay | Bioorg Med Chem Lett 21: 6451-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.084 BindingDB Entry DOI: 10.7270/Q26W9BG8 | |||||||||||
More data for this Ligand-Target Pair |