Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50095114 (4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-benzoyl]-[1,4'...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Binding affinity at human cloned acetylcholine receptor M2 in CHO cells. | Bioorg Med Chem Lett 10: 2727-30 (2000) BindingDB Entry DOI: 10.7270/Q2V40TGZ | |||||||||||
More data for this Ligand-Target Pair |