Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M3 (RAT) | BDBM50034625 (Aceclidine | Acetic acid 1-aza-bicyclo[2.2.2]oct-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | PubMed | 22.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by PDSP Ki Database | J Pharmacol Exp Ther 279: 1335-44 (1996) BindingDB Entry DOI: 10.7270/Q2XG9PPG | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (RAT) | BDBM50034625 (Aceclidine | Acetic acid 1-aza-bicyclo[2.2.2]oct-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by PDSP Ki Database | J Pharmacol Exp Ther 279: 1335-44 (1996) BindingDB Entry DOI: 10.7270/Q2XG9PPG | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Mus musculus) | BDBM50034625 (Aceclidine | Acetic acid 1-aza-bicyclo[2.2.2]oct-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
The University of Toledo Curated by ChEMBL | Assay Description Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell line | J Med Chem 40: 1230-46 (1997) Article DOI: 10.1021/jm960467d BindingDB Entry DOI: 10.7270/Q28916HS | |||||||||||
More data for this Ligand-Target Pair |