Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50241913 (CHEMBL499519 | GNF-PF-5618 | nocardimicin B) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Pharma Corporation Curated by ChEMBL | Assay Description Binding affinity to human muscarinic M4 receptor expressed in insect Sf9 cells | J Nat Prod 68: 1061-5 (2005) Article DOI: 10.1021/np050091j BindingDB Entry DOI: 10.7270/Q2R21155 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50241913 (CHEMBL499519 | GNF-PF-5618 | nocardimicin B) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Pharma Corporation Curated by ChEMBL | Assay Description Binding affinity to human muscarinic M4 receptor expressed in insect Sf9 cells | J Nat Prod 68: 1061-5 (2005) Article DOI: 10.1021/np050091j BindingDB Entry DOI: 10.7270/Q2R21155 | |||||||||||
More data for this Ligand-Target Pair |