Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
NUAK family SNF1-like kinase 1 (Homo sapiens (Human)) | BDBM50243878 (3-(1H-Indol-3-yl)-4-(3,4,5-trimethoxyphenyl)-1,5-d...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Eberhard-Karls University Curated by ChEMBL | Assay Description Inhibition of human recombinant ARK5 | J Med Chem 51: 3814-24 (2008) Article DOI: 10.1021/jm8001185 BindingDB Entry DOI: 10.7270/Q2057FQS | |||||||||||
More data for this Ligand-Target Pair |