Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078966 (1-Benzo[b]thiophen-5-yl-3-{1-[3-(3-isopropyl-ureid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair |