Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50246613 ((R)-N-(4-hydroxybenzyl)-5-(2-acetylguanidino)-2-(2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Regensburg Curated by ChEMBL | Assay Description Displacement of [3H]propionyl-pNPY from neuropeptide Y1 receptor in human SK-N-MC cells | J Med Chem 51: 8168-72 (2008) Article DOI: 10.1021/jm801018u BindingDB Entry DOI: 10.7270/Q2WM1D8T | |||||||||||
More data for this Ligand-Target Pair |